MALEGRA PRO-100

In the treatment of erectile dysfunction (ED), combining maximum efficacy with a fast onset of action is crucial. MALEGRA PRO-100 is an advanced generic containing the maximum standard dose of Sildenafil Citrate (100 mg) in a sublingual tablet form (for dissolving under the tongue). This form ensures ultra-fast absorption and is ideal for men who require a guaranteed and quick effect.

What is MALEGRA PRO-100?

MALEGRA PRO-100 is an oral medication containing 100 mg of Sildenafil. The distinctive feature of the "Pro" version is the sublingual form (dissolvable tablets).

1. Indication and target dosage

The 100 mg Sildenafil dose is the maximum recommended daily dose for ED treatment. MALEGRA PRO-100 is suitable for men who:

• Did not achieve a sufficient therapeutic response from the 50 mg dose.

• Have moderate or severe ED, where 100 mg is necessary for a guaranteed effect.

• Require the fastest possible onset of action.

2. Advantage of the sublingual form

The sublingual form (dissolving under the tongue) provides:

• Ultra-Fast Effect: Sildenafil is absorbed directly into the bloodstream through the oral mucosa, bypassing the liver. The effect can start in as little as 15–25 minutes, which is significantly faster than a regular tablet.

• Independence from the Stomach: Food intake hardly affects the speed of absorption, helping to maintain spontaneity.

• Convenience: The tablet does not need to be washed down with water, making intake discreet.

Detailed mechanism of action of MALEGRA PRO-100

The mechanism of action of MALEGRA PRO-100 is based on Sildenafil 100 mg being a potent PDE5 enzyme inhibitor.

1. Trigger: Sexual arousal causes the release of nitric oxide (NO).

2. Erectile Cycle: NO stimulates the formation of cyclic GMP (cGMP), which relaxes the smooth muscles of the penile blood vessels, ensuring a powerful blood flow.

3. Blockade: Sildenafil blocks the PDE5 enzyme that degrades cGMP. Blocking this enzyme allows cGMP to persist longer, manifold enhancing the natural blood flow and ensuring a stable, firm erection.

Key takeaway: MALEGRA PRO-100 enhances the physiological response but does not cause an erection without sexual arousal.

Instructions for using MALEGRA PRO-100

Strict adherence to the instructions is necessary for safety and maximum speed of action.

1. Dosage and method of intake

• Dosage: 100 mg (one tablet) – is the maximum daily dose. It is strictly prohibited to exceed 100 mg within 24 hours.

• Initial Dose: If you are trying Sildenafil for the first time, it is recommended to start with half a tablet (50 mg) to assess tolerability. The MALEGRA PRO-100 tablet is easily scored for splitting.

• Method: Place the tablet under the tongue and hold until fully dissolved. Do not swallow it whole to preserve the advantage of fast absorption.

• Timing: Take 15–25 minutes before planned activity.

2. Influence of food and alcohol

• Food: Taking it on an empty stomach guarantees the fastest effect.

• Alcohol: Strictly not recommended to combine Sildenafil intake with alcohol, as this enhances the vasodilating effect, increasing the risk of headaches and hypotension.

Critical contraindications for MALEGRA PRO-100

The risk of side effects and interactions at the 100 mg dose is high.

• Interaction with Nitrates: Absolutely forbidden! Taking MALEGRA PRO-100 with any form of organic nitrates (Nitroglycerin) or nitric oxide donors ("poppers") causes a life-threatening drop in blood pressure.

• Severe Cardiovascular Diseases: Recent heart attack or stroke (within 6 months), unstable angina, severe heart failure.

• Blood Pressure: Persistent hypotension (pressure < 90/50 mmHg) or uncontrolled hypertension.

• Liver and Kidneys: Severe hepatic or renal failure.

• Eyes: Hereditary degenerative retinal diseases (retinitis pigmentosa).

Side effects of MALEGRA PRO-100

At the 100 mg dose, side effects are more frequent and can be more pronounced than at 50 mg.

• Common: Headache (the most frequent effect), facial flushing, nasal congestion.

• Less Common: Visual disturbances (temporary change in color perception, "blue haze"), dyspepsia, dizziness.

Immediate medical attention is required for: An erection that lasts longer than 4 hours (priapism), or sudden loss of vision/hearing.

Professional advice on using MALEGRA PRO-100

1. Speed and Spontaneity: The sublingual form makes MALEGRA PRO-100 an ideal choice for situations requiring fast and discreet intake, without the need to find water. It is "the date pill."

2. Dosing Flexibility: The tablet can be split into two parts (50 mg) or even four (25 mg), allowing you to find the minimum effective dose, minimizing side effects.

3. Blood Pressure Control: The rapid absorption of Sildenafil can lead to a more sudden, though transient, change in blood pressure. Be cautious when standing up abruptly.

MALEGRA PRO-100: Extended Q&A section

• How much faster is MALEGRA PRO-100 than a regular tablet? Thanks to sublingual absorption, the effect can start 20–40 minutes faster than if swallowed.

• How long does MALEGRA PRO-100 last? The duration of action of Sildenafil 100 mg averages 4-6 hours. The release form affects speed but not duration.

• What is the difference between MALEGRA PRO-100 and MALEGRA PRO-50? The difference is only in the dosage of the active substance. MALEGRA PRO-100 is stronger, but MALEGRA PRO-50 is safer for starting.

• Can MALEGRA PRO-100 be swallowed? Technically yes, but this eliminates the main advantage of the drug—speed. If swallowed, it will work like a regular tablet in 45-60 minutes.